About: Characterisation of the binding of [3H]WAY-100635, a novel 5-hydroxytryptamine1A receptor antagonist, to rat brain

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About: Characterisation of the binding of [3H]WAY-100635, a novel 5-hydroxytryptamine1A receptor antagonist, to rat brain Goto Sponge Distinct Permalink

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scientific article published on 01 June 1995

Attributes	Values
rdf:type	Item
description	wetenschappelijk artikel (nl) наукова стаття, опублікована в червні 1995 (uk) artículu científicu espublizáu en xunu de 1995 (ast) scientific article published on 01 June 1995 (en)
publication date	wds:Q72261240-0EABEB9E-1140-47E8-98D0-3F93AD8C3FD0
publication date	1995-06-01 00:00:00Z (xsd:dateTime)
author name string	wds:Q72261240-07D3B157-2043-4446-9DFC-069A748966BF wds:Q72261240-2E270C62-B85B-4DD7-A21A-A08DD0676D74 wds:Q72261240-392FC3B9-E423-47CF-B7E5-F8D772DAAAD9 wds:Q72261240-D02FD773-727E-45D4-ADB6-229D4DFF1CC8 wds:Q72261240-F0030D07-D57F-4FFB-A451-138ACE92EFD8
author name string	N Evans C Ennis M C Minchin Y Reilly X Khawaja
rdfs:label	Characterisation of the binding of [3H]WAY-100635, a novel 5-hydroxytryptamine1A receptor antagonist, to rat brain (en) Characterisation of the binding of [3H]WAY-100635, a novel 5-hydroxytryptamine1A receptor antagonist, to rat brain (nl)
skos:prefLabel	Characterisation of the binding of [3H]WAY-100635, a novel 5-hydroxytryptamine1A receptor antagonist, to rat brain (en) Characterisation of the binding of [3H]WAY-100635, a novel 5-hydroxytryptamine1A receptor antagonist, to rat brain (nl)
name	Characterisation of the binding of [3H]WAY-100635, a novel 5-hydroxytryptamine1A receptor antagonist, to rat brain (en) Characterisation of the binding of [3H]WAY-100635, a novel 5-hydroxytryptamine1A receptor antagonist, to rat brain (nl)
title	wds:Q72261240-76E7B270-A974-44D9-968D-218AD70E0F23
title	Characterisation of the binding of [3H]WAY-100635, a novel 5-hydroxytryptamine1A receptor antagonist, to rat brain (en)
page(s)	wds:Q72261240-315A6B73-23D3-43A0-ADE6-E10423A8D143
page(s)	2716-2726
instance of	wds:Q72261240-0F4999C9-97CF-49D1-9885-1C4DEF619975
instance of	scholarly article
PubMed ID	wds:Q72261240-1C758E01-B602-41E4-A8DB-FAAB4AA9ABB1
PubMed ID	http://rdf.ncbi.nlm.nih.gov/pubchem/reference/7760052
PubMed ID	7760052
published in	wds:Q72261240-6B26E98E-27F2-4735-8831-E8F416E2F0D1
published in	Journal of Neurochemistry
issue	wds:Q72261240-7AD24A49-7C2F-4E92-BCEE-3366B1FEEC23
volume	wds:Q72261240-AE7D4B90-1FE5-493F-8DE2-D9335C0D25C3
issue	6
volume	64
DOI	wds:Q72261240-64F4A1E2-2A2A-4067-AEA0-4303AB584063
DOI	http://dx.doi.org/10.1046/J.1471-4159.1995.64062716.X
DOI	10.1046/J.1471-4159.1995.64062716.X
is about of	https://www.wikidata.org/wiki/Special:EntityData/Q72261240
is cites work of	5-HT7 receptors mediate serotonergic effects on light-sensitive suprachiasmatic nucleus neurons. Measurement of serotonin 5-HT1A receptor binding using positron emission tomography and [carbonyl-(11)C]WAY-100635-considerations on the validity of cerebellum as a reference region Effects of selective 5-HT1A receptor antagonists on regional serotonin synthesis in the rat brain: an autoradiographic study with alpha-[14C]methyl-L-tryptophan Receptor binding characteristics of [3H]NAD-299, a new selective 5-HT1A receptor antagonist Pharmacological characterization of recombinant human 5-hydroxytryptamine1A receptors using a novel antagonist radioligand, [3H]WAY-100635. Characterisation of the appearance of radioactive metabolites in monkey and human plasma from the 5-HT1A receptor radioligand, [carbonyl-11C]WAY-100635--explanation of high signal contrast in PET and an aid to biomathematical modelling. Autoradiographic localization of 5-HT1A receptors in the post-mortem human brain using [3H]WAY-100635 and [11C]way-100635 Modulation of the firing activity of noradrenergic neurones in the rat locus coeruleus by the 5-hydroxtryptamine system Control of dorsal raphe serotonergic neurons by the medial prefrontal cortex: Involvement of serotonin-1A, GABA(A), and glutamate receptors. Sustained blockade of neurokinin-1 receptors enhances serotonin neurotransmission Respiratory and cardiovascular effects of the mu-opioid receptor agonist [Lys7]dermorphin in awake rats Autoradiographic distribution of serotonin transporters and receptor subtypes in human brain Long-term antidepressant treatments result in a tonic activation of forebrain 5-HT1A receptors. Fluoro analogs of WAY-100635 with varying pharmacokinetics properties Derivatives of WAY 100635 as potential imaging agents for 5-HT1A receptors: syntheses, radiosyntheses, and in vitro and in vivo evaluation. Quantitative analysis of [carbonyl-11C]WAY-100635 PET studies Estrogen modulates 5-HT(1A) agonist inhibition of lordosis behavior but not binding of [(3)H]-8-OH-DPAT. Effect of the selective 5-HT1A receptor antagonist WAY 100635 on the inhibition of e.p.s.ps produced by 5-HT in the CA1 region of rat hippocampal slices Diabetes attenuates the antidepressant-like effect mediated by the activation of 5-HT1A receptor in the mouse tail suspension test The PET radioligand [11C]MePPEP binds reversibly and with high specific signal to cannabinoid CB1 receptors in nonhuman primate brain Radioligands for the study of brain 5-HT1A receptors in vivo. Acute and chronic tryptophan depletion differentially regulate central 5-HT1A and 5-HT 2A receptor binding in the rat. Mutation in a protein kinase C phosphorylation site of the 5-HT1A receptor preferentially attenuates Ca2+ responses to partial as opposed to higher-efficacy 5-HT1A agonists In vivo intrinsic efficacy of the 5-HT1A receptor antagonists NAD-299, WAY-100,635 and (S)-(-)-UH-301 at rat brain monoamine receptors. Measurement of 5-HT(1A) receptor density and in-vivo binding parameters of [(18)F]mefway in the nonhuman primate. Evaluation of serotonin 5-HT(1A) receptors in rodent models using [¹⁸F]mefway PET. Distribution of the 5-HT(1A) receptor antagonist [ (18)F]FPWAY in blood and brain of the rat with and without isoflurane anesthesia. Pindolol augmentation of antidepressant treatment: recent contributions from brain imaging studies A review of the neuroprotective properties of the 5-HT1A receptor agonist repinotan HCl (BAYx3702) in ischemic stroke. Enhancement of serotonergic and noradrenergic neurotransmission in the rat hippocampus by sustained administration of bupropion. Metal ion and guanine nucleotide modulations of agonist interaction in G-protein-coupled serotonin1A receptors from bovine hippocampus. The 5-HT1A receptor agonist BAY x 3702 prevents staurosporine-induced apoptosis. Effects of WAY 100635 and (-)-5-Me-8-OH-DPAT, a novel 5-HT1A receptor antagonist, on 8-OH-DPAT responses. Juvenile stress attenuates the dorsal hippocampal postsynaptic 5-HT1A receptor function in adult rats. Characteristics of binding of [3H]WAY100635 to rat hippocampal membranes. Comparative assessment of (18) F-Mefway as a serotonin 5-HT1A receptor PET imaging agent across species: Rodents, nonhuman primates, and humans Measuring endogenous 5-HT release by emission tomography: promises and pitfalls Contractile effects of 5-hydroxytryptamine and 5-carboxamidotryptamine in the equine jejunum GR46611 potentiates 5-HT1A receptor-mediated locomotor activity in the guinea pig. Preclinical evaluation and quantification of [¹⁸F]MK-9470 as a radioligand for PET imaging of the type 1 cannabinoid receptor in rat brain. Facilitation by 8-OH-DPAT of passive avoidance performance in rats after inactivation of 5-HT(1A) receptors Electroconvulsive shock increases tachykinin NK(1) receptors, but not the encoding mRNA, in rat cortex. Presynaptic selectivity of a ligand for serotonin 1A receptors revealed by in vivo PET assays of rat brain
is cites work of	wds:Q48260745-8F15E430-9FB1-458B-A6F4-22A2A53431B9 wds:Q48087754-93449BD8-7E2B-440F-ADDF-ADCF40246DAA wds:Q43182815-876AD413-E842-4E08-A224-75E033C936CC wds:Q48323277-E073DDEB-B5FD-409B-8807-60F3BF796935 wds:Q48708666-7A422B77-7558-432B-A095-2DEB5F5AD978 wds:Q37776154-BE37A70E-BF2F-4865-8C43-8EBADDECE2CC wds:Q48473239-DB3F4B2D-5C7B-42A2-9545-BE074E7ED680 wds:Q28239230-F21FFE8B-2CE9-470A-B2B2-5894CC9CDA3A wds:Q30498723-7D4B89BB-4652-41C9-B659-082C42241BA2 wds:Q33995061-F31EF4CB-74C3-4A0B-AF33-5A4BDD01BDC0 wds:Q48968624-962E75CE-99A8-497F-8F5C-FBC2A35FC9FE wds:Q34483298-A1CB4B1C-2B76-48C8-B67F-854BF41BF2C2 wds:Q40855928-8194F0CF-647E-47D3-A3BE-4588E7B7417E wds:Q48435371-360B8DD4-FF8C-4B66-877D-3858C0CFAA31 wds:Q44662310-826B321A-BC39-429F-BFE2-C364BEB6CE23

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